Re: ORGLIST: Amination of a chlorobenzyl

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From: Uno Mäeorg (uno$##$chem.ut.ee)
Date: Thu Nov 29 2007 - 16:04:16 EST

Previous message: Alexey Gromov: "Re: ORGLIST: imide synthesis maleamic acid"
Maybe in reply to: Mar Quesada: "ORGLIST: Amination of a chlorobenzyl"

Hi Mar,

You could make the corresponding boronic acid or triaryl bismuthane from the ArHal derivative and use the simple Cu-catalysis in presence of TEA and in DCM for amination.

Regards

Uno

At 03:43 PM 11/29/2007, Mar Quesada wrote:

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Hi all

Any ideas of how to aminate the chloro position of a phenyl ring? I know you could use Buchwald, but it might be tricky, so any other suggestions?

Thank you

Mar

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Previous message: Alexey Gromov: "Re: ORGLIST: imide synthesis maleamic acid"
Maybe in reply to: Mar Quesada: "ORGLIST: Amination of a chlorobenzyl"

Date view	Thread view	Subject view	Author view	Attachment view

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